Affinity DataKi: 4.20nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition constants against ATP substrate site of M-2 (kidney form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 44.3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition constants against Met (L-methionine)P substrate site of M-T (Novikoff Ascitic Hepatoma form) variant of rat Methionine adenosyltransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity measured on human cytochrome P450 2C9 (CYP2C9) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Inhibition of purified CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity measured on human cytochrome P450 2C9 (CYP2C9) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of human cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity towards cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 656nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Competitive inhibition of CYP2C8 in human liver microsomes assessed as paclitaxel 6-hydroxylation after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Mechanism based inhibition of human cytochrome P450 2C8 measured by paclitaxel hydroxylation using a recombinant systemMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+3nMAssay Description:Binding affinity to CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Mechanism based inhibition of human cytochrome P450 2C8 measured by paclitaxel hydroxylation using a recombinant systemMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity was measured on Cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Biphasic inhibition of CYP2C8 in human liver microsomes assessed as montelukast 36-hydroxylation after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+3nMAssay Description:Inhibition of reconstituted CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity towards cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity measured on human cytochrome P450 2C9 (CYP2C9) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity measured on human cytochrome P450 2C9 (CYP2C9) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity towards cytochrome P450 2C9More data for this Ligand-Target Pair